Design, synthesis, and SAR of a novel pyrazinone series with non-nucleoside HIV-1 reverse transcriptase inhibitory activity.
نویسندگان
چکیده
A series of novel pyrazinones designed as non-nucleoside reverse transcriptase inhibitors (NNRTIs) was synthesized and their anti-HIV structure-activity relationship (SAR) was studied.
منابع مشابه
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ورودعنوان ژورنال:
- Journal of medicinal chemistry
دوره 48 6 شماره
صفحات -
تاریخ انتشار 2005